Title: A facile diversity-Oriented Synthesis of Imidazo[1,2-a]pyrazinones via Gold-Catalyzed Regioselective Heteroannulation of Propynylaminopyrazinones
Authors: Vachhani, Dipakkumar
Modha, Sachinkumar
Sharma, Abhishek
Van der Eycken, Erik # ×
Issue Date: Jan-2013
Publisher: Pergamon Press
Series Title: Tetrahedron vol:69 issue:1 pages:359-365
Abstract: A gold-catalyzed regioselective heteroannulation strategy has been developed for the concise
and efficient synthesis of imidazo[1,2-a]pyrazinones. The protocol allows the introduction of
diversity via the application of substituted propargyl amines or via Suzuki-coupling of the
generated imidazo[1,2-a]pyrazinones with various (het)aryl boronic acids.
ISSN: 0040-4020
Publication status: published
KU Leuven publication type: IT
Appears in Collections:Molecular Design and Synthesis
× corresponding author
# (joint) last author

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